Compound | Asinex Identifier a | Structure | Serum PON1 IC50 (µM) b | Purified PON1 | |
---|---|---|---|---|---|
% Inhibition c | IC50 (µM) d | ||||
2HQ | N/A | 7.9 | 84 | 4.4 | |
1 | ASN 08910296 | 8.5 | 90 | 10.6 | |
2 | ASN 08912428 | 18.6 | 13 | n.d. e | |
3 | BAS 09529674 | 15.3 | 103 | 0.76 | |
4 | BAS 01369653 | 10.3 | 90 | 5.3 | |
5 | BAS 09683917 | 21.8 | -2 | n.d. | |
6 | BAS 09683916 | 26.6 | 6 | n.d. | |
7 | BAS 03551158 | 12.5 | 103 | 0.42 | |
8 | ASN 05298740 | 13.2 | 12 | n.d. | |
9 | BAS 05307909 | 14.9 | 70 | n.d. | |
10 | BAS 02915353 | 18.4 | 19 | n.d. | |
11 | BAS 09588626 | 20.6 | 92 | 4.8 | |
12 | BAS 01814176 | 21.1 | 18 | n.d. |