Table 3:
Comparison of EC
50
(Agonists) and IC
50
(Antago-nists) for m
3
Muscarinic Receptor by NFAT-RE- and SRE- Luciferase Reporter Assays
agonist
NFAT-RE, EC
50
(M)
SRE, EC
50
(M)
muscarine chloride
8.3 × 10
-9
2.8 ×10
-8
carbachol
3.6 × 10
-8
1.1 × 10
-7
pilocarpine
2.0 × 10
-7
5.2 × 10
-7